Acetazolamide Ext-rel Caps

— THERAPEUTIC CATEGORIES —
  • Glaucoma

Acetazolamide Ext-rel Caps Generic Name & Formulations

General Description

Acetazolamide 500mg.

Pharmacological Class

Carbonic anhydrase inhibitor.

How Supplied

Contact supplier

Acetazolamide Ext-rel Caps Indications

Indications

Adjunct in open-angle glaucoma.

Acetazolamide Ext-rel Caps Dosage and Administration

Adult

500mg twice daily.

Children

Not established.

Acetazolamide Ext-rel Caps Contraindications

Contraindications

Hypokalemia. Hyponatremia. Severe renal, hepatic, or adrenocortical impairment. Hyperchloremic acidosis. Cirrhosis. Chronic noncongestive angle-closure glaucoma. Sulfonamide allergy.

Acetazolamide Ext-rel Caps Boxed Warnings

Not Applicable

Acetazolamide Ext-rel Caps Warnings/Precautions

Warnings/Precautions

Respiratory impairment. Renal calcium calculi. Diabetes. Gout. Test blood periodically in chronic use. Pregnancy (Cat.C). Nursing mothers: not recommended.

Acetazolamide Ext-rel Caps Pharmacokinetics

See Literature

Acetazolamide Ext-rel Caps Interactions

Interactions

May inhibit renal excretion of basic drugs and promote excretion of acidic drugs. May increase salicylate toxicity (acidosis). Hypokalemia with corticosteroids, potassium wasting diuretics.

Acetazolamide Ext-rel Caps Adverse Reactions

Adverse Reactions

Anorexia, drowsiness, confusion, malaise, depression, GI distress, paresthesias, tinnitus, acidosis, initial hypokalemia, hyperuricemia, transient myopia; renal calculi, nephrotoxicity, hepatic dysfunction, blood dyscrasias, rash, fever, photosensitivity (rare).

Acetazolamide Ext-rel Caps Clinical Trials

See Literature

Acetazolamide Ext-rel Caps Note

Notes

Formerly known under the brand name Diamox Sequels.

Acetazolamide Ext-rel Caps Patient Counseling

See Literature