Estazolam

— THERAPEUTIC CATEGORIES —
  • Sleep-wake disorders

Estazolam Generic Name & Formulations

General Description

Estazolam 1mg, 2mg; scored tabs.

Pharmacological Class

Benzodiazepine.

How Supplied

Contact supplier.

Estazolam Indications

Indications

Short-term treatment of insomnia.

Estazolam Dosage and Administration

Adult

Initially 1mg at bedtime. May increase to 2mg nightly. Small or debilitated elderly: initially 0.5mg.

Children

<18yrs: not recommended.

Estazolam Contraindications

Contraindications

Concomitant ketoconazole, itraconazole. Pregnancy (Cat.X).

Estazolam Boxed Warnings

Not Applicable

Estazolam Warnings/Precautions

Warnings/Precautions

Drug or alcohol abuse. Suicidal tendencies. Depression. Renal, hepatic, or respiratory impairment. Avoid abrupt cessation after prolonged use. Elderly. Debilitated. Nursing mothers: not recommended.

Estazolam Pharmacokinetics

See Literature

Estazolam Interactions

Interactions

Potentiates CNS depression with alcohol, other CNS depressants. Caution with CYP3A inhibitors (eg, nefazodone, fluvoxamine, cimetidine, diltiazem, isoniazid, other macrolides): consider dose reduction.

Estazolam Adverse Reactions

Adverse Reactions

CNS depression, complex sleep-related behaviors (eg, sleep-driving), hypokinesia, dizziness, incoordination, confusion, constipation, anxiety, paradoxical excitement; anaphylaxis, angioedema.

Estazolam Clinical Trials

See Literature

Estazolam Note

Notes

Formerly known under the brand name Prosom.

Estazolam Patient Counseling

See Literature