Betimol

— THERAPEUTIC CATEGORIES —
  • Glaucoma

Betimol Generic Name & Formulations

General Description

Timolol (as hemihydrate) 0.25%, 0.5%; oph. soln; contains benzalkonium chloride.

Pharmacological Class

Noncardioselective beta-blocker.

How Supplied

Soln—5mL, 10mL, 15mL

Manufacturer

Betimol Indications

Indications

Open-angle glaucoma.

Betimol Dosage and Administration

Adult

1 drop twice daily.

Children

Not recommended.

Betimol Contraindications

Contraindications

Overt heart failure. Cardiogenic shock. Sinus bradycardia. 2nd- or 3rd-degree AV block. Asthma. Severe COPD.

Betimol Boxed Warnings

Not Applicable

Betimol Warnings/Precautions

Warnings/Precautions

Discontinue if heart failure develops and prior to surgery. Not for use as sole agent in narrow-angle glaucoma. Avoid abrupt cessation. Cerebrovascular insufficiency. Diabetes. COPD. Bronchospastic disease. May mask signs of hypoglycemia, thyrotoxicosis. Myasthenia gravis. Bacterial keratitis. Measure IOP after 4 wks of treatment. Pregnancy (Cat.C). Nursing mothers: not recommended.

Betimol Pharmacokinetics

See Literature

Betimol Interactions

Interactions

May potentiate systemic β-blockers, reserpine. May cause conduction defects with calcium channel blockers, digitalis. May antagonize β-agonists. May block epinephrine.

Betimol Adverse Reactions

Adverse Reactions

Ocular irritation, eyelid erythema, conjunctival injection, headache, epiphora, photophobia. Systemic β-blocking effects (bradycardia, arrhythmias, hypotension, bronchospasm, heart failure).

Betimol Clinical Trials

See Literature

Betimol Note

Not Applicable

Betimol Patient Counseling

See Literature