Salsalate

— THERAPEUTIC CATEGORIES —
  • Arthritis/rheumatic disorders

Salsalate Generic Name & Formulations

General Description

Salsalate 500mg, 750mg; scored tabs.

Pharmacological Class

Salicylate.

See Also

    How Supplied

    Contact supplier.

    Salsalate Indications

    Indications

    Rheumatoid arthritis. Osteoarthritis.

    Salsalate Dosage and Administration

    Adult

    3g daily in divided doses.

    Children

    Not recommended.

    Salsalate Contraindications

    Contraindications

    Varicella or influenza in teenagers. 3rd trimester pregnancy. Aspirin allergy. Coronary artery bypass graft surgery.

    Salsalate Boxed Warnings

    Not Applicable

    Salsalate Warnings/Precautions

    Warnings/Precautions

    Advanced renal disease: not recommended. Impaired renal or hepatic function. Hypertension. Heart failure. Edema. Bleeding disorders. Monitor blood, liver, renal function with chronic use. Peptic ulcer. Gastritis. Diabetes. Elderly. Debilitated. Pregnancy (Cat.C). Nursing mothers: not recommended.

    Salsalate Pharmacokinetics

    See Literature

    Salsalate Interactions

    Interactions

    PABA may increase serum levels. May potentiate anticoagulants, hypoglycemics, methotrexate. Urinary alkalinizers, antacids, corticosteroids may increase excretion. May antagonize uricosurics and spironolactone.

    Salsalate Adverse Reactions

    Adverse Reactions

    Salicylism, tinnitus, nausea, dyspepsia, GI bleed, hearing loss, rash (discontinue if occurs). See literature re: risk of cardiovascular events.

    Salsalate Clinical Trials

    See Literature

    Salsalate Note

    Notes

    Formerly known under the brand names Disalcid, Salflex.

    Salsalate Patient Counseling

    See Literature